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Uchanganuzi wa Utendaji wa Dawa unaolenga Lengo

Uchanganuzi wa utendaji wa dawa unaolenga lengo (TMDD) ni mfumo wa kiufundi unaoelezea farmakokinetiki isiyo sawia inayotokana na kufungamana kwa dawa na kipokezi au protini lengo. Uliandaliwa na Mager na Jusko mwaka 2001, TMDD unaelezea msafara unaofikia kikomo, muda wa nusu unaotegemea kipimo, na mabadiliko yanayotegemea muda katika viwango vya dawa mwilini vinavyoonekana kwa tiba za protini na baadhi ya dawa za molekuli ndogo.

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Vyanzo

  1. Mager, D. E., & Jusko, W. J. (2001). General pharmacokinetic model for drugs exhibiting target-mediated drug disposition. Journal of Pharmacokinetics and Pharmacodynamics, 28(6), 507-532. DOI: 10.1023/A:1014414520282
  2. Levy, G. (2004). Carrier-mediated active transport: pharmacokinetic consequences and examples in humans. Clinical Pharmacokinetics, 37(6), 429-445. link

Jinsi ya kunukuu ukurasa huu

ScholarGate. (2026, June 3). Target-Mediated Drug Disposition (TMDD). ScholarGate. https://scholargate.app/sw/pharmacology/target-mediated-drug-disposition

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ScholarGateTarget-Mediated Drug Disposition (Target-Mediated Drug Disposition (TMDD)). Imepatikana 2026-06-19 kutoka https://scholargate.app/sw/pharmacology/target-mediated-drug-disposition · Seti ya data: https://doi.org/10.5281/zenodo.20539026