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Fator de Similaridade f1/f2 para Dissolução×Cinética de Michaelis-Menten×
ÁreaFarmacologiaFarmacologia
FamíliaProcess / pipelineProcess / pipeline
Ano de origem19961913
Autor originalJames Moore and Hector FlannerLeonor Michaelis and Maud Menten
Tiposimilarity testingmechanistic model
Fonte seminalMoore, J. W., & Flanner, H. H. (1996). Mathematical comparison of dissolution profiles. Pharmaceutical Technology, 20(6), 64-74. link ↗Michaelis, L., & Menten, M. L. (1913). Die Kinetik der Invertinwirkung. Biochemische Zeitschrift, 49, 333-369. link ↗
Outros nomesf1, f2, similarity factorMM kinetics, Michaelis constant, Vmax
Relacionados32
ResumoThe f1 and f2 factors are dimensionless statistical measures developed by Moore and Flanner to quantify the similarity between two dissolution profiles. Adopted by regulatory agencies (FDA, EMA) as the gold standard for comparing dissolution curves, these factors enable rapid assessment of whether formulation changes significantly impact drug release.Michaelis-Menten kinetics describes the rate of enzyme-catalyzed reactions as a function of substrate concentration. Developed by Leonor Michaelis and Maud Menten in 1913, this foundational framework models enzyme catalysis through the rapid-equilibrium approximation and enables prediction of drug metabolism rates in pharmacokinetics.
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ScholarGateComparar métodos: Dissolution f1/f2 Similarity · Michaelis-Menten Kinetics. Recuperado em 2026-06-20 de https://scholargate.app/pt/compare