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Schildova analiza×Populacijsko farmakodinamičko modeliranje×
PodručjeFarmakologijaFarmakologija
ObiteljProcess / pipelineProcess / pipeline
Godina nastanka19471992
TvoracHenry SchildLewis Sheiner and Stephen Roush
Vrstaantagonism quantificationdose-response modeling
Temeljni izvorSchild, H. O. (1947). pA, a new scale for the measurement of drug antagonism. Journal of Physiology, 106(3), 337-357. DOI ↗Dahlström, B., & Nyberg, L. (1993). Population pharmacokinetics and pharmacodynamics. Clinical Pharmacokinetics, 24(1), 45-57. link ↗
Drugi naziviSchild plot, pA2PopPD, population PD, hierarchical PD modeling
Srodne33
SažetakSchild analysis is a quantitative method for characterizing competitive receptor antagonism developed by Henry Schild in 1947. It uses dose-response curves in the presence and absence of antagonist to estimate the antagonist affinity constant (pA2), enabling standardized comparison of antagonist potency across drugs and experimental systems.Population pharmacodynamic (PopPD) modeling integrates pharmacokinetics with individual dose-response relationships across patient populations to characterize drug efficacy and tolerability. Pioneered by Lewis Sheiner and colleagues, PopPD accounts for inter-individual variability in drug effects and enables rational dose optimization and response prediction.
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ScholarGateUsporedite metode: Schild Analysis · Population Pharmacodynamics. Preuzeto 2026-06-18 s https://scholargate.app/hr/compare