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Process / pipelineBiopharmaceutics

Kipimo cha Upenyezaji wa Seli za Caco-2

Kipimo cha Caco-2 ni mfumo wa mfano wa in vitro unaotumia monola ya seli za kansa ya utumbo mpana wa binadamu kuchuja upenyezaji wa dawa kwenye utumbo. Iliyotengenezwa na Hidalgo na washirika mnamo 1989, seli za Caco-2 hujitofautisha na kuwa kizuizi cha epitheliamu kinachofanana na utando wa utumbo, kuwezesha tathmini ya haraka ya uwezo wa dawa kufyonzwa na utambuzi wa usafirishaji unaosimamiwa na vichukuzi.

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Vyanzo

  1. Hidalgo, I. J., Raub, T. J., & Borchardt, R. T. (1989). Characterization of the human colon carcinoma cell line (Caco-2) as a model system for intestinal epithelial permeability. Gastroenterology, 96(3), 736-749. DOI: 10.1016/S0016-5085(89)80072-1
  2. Artursson, P. (1990). Epithelial transport of drugs in cell culture. I: A model for studying the passive diffusion of drugs over intestinal absorptive (Caco-2) cells. Journal of Pharmaceutical Sciences, 79(6), 476-482. DOI: 10.1002/jps.2600790604

Jinsi ya kunukuu ukurasa huu

ScholarGate. (2026, June 3). Caco-2 Cell Permeability Assay. ScholarGate. https://scholargate.app/sw/pharmacology/caco-2-permeability

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Imerejelewa na

ScholarGateCaco-2 Permeability (Caco-2 Cell Permeability Assay). Imepatikana 2026-06-17 kutoka https://scholargate.app/sw/pharmacology/caco-2-permeability · Seti ya data: https://doi.org/10.5281/zenodo.20539026