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Modelarea Farmacodinamică Populațională×Analiza Schild×
DomeniuFarmacologieFarmacologie
FamilieProcess / pipelineProcess / pipeline
Anul apariției19921947
Autorul originalLewis Sheiner and Stephen RoushHenry Schild
Tipdose-response modelingantagonism quantification
Sursa seminalăDahlström, B., & Nyberg, L. (1993). Population pharmacokinetics and pharmacodynamics. Clinical Pharmacokinetics, 24(1), 45-57. link ↗Schild, H. O. (1947). pA, a new scale for the measurement of drug antagonism. Journal of Physiology, 106(3), 337-357. DOI ↗
Denumiri alternativePopPD, population PD, hierarchical PD modelingSchild plot, pA2
Înrudite33
RezumatPopulation pharmacodynamic (PopPD) modeling integrates pharmacokinetics with individual dose-response relationships across patient populations to characterize drug efficacy and tolerability. Pioneered by Lewis Sheiner and colleagues, PopPD accounts for inter-individual variability in drug effects and enables rational dose optimization and response prediction.Schild analysis is a quantitative method for characterizing competitive receptor antagonism developed by Henry Schild in 1947. It uses dose-response curves in the presence and absence of antagonist to estimate the antagonist affinity constant (pA2), enabling standardized comparison of antagonist potency across drugs and experimental systems.
ScholarGateSet de date
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  2. 2 Surse
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  1. v1
  2. 2 Surse
  3. PUBLISHED

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ScholarGateCompară metode: Population Pharmacodynamics · Schild Analysis. Preluat la 2026-06-18 de pe https://scholargate.app/ro/compare