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Livrarea Medicamentelor Lipozomale×Formulare prin dispersie solidă×
DomeniuFarmacologieFarmacologie
FamilieProcess / pipelineProcess / pipeline
Anul apariției19651971
Autorul originalAlec BanghamWilliam Chiou and Solomon Riegelman
Tipformulation technologysolubility enhancement
Sursa seminalăBangham, A. D., Standish, M. M., & Watkins, J. C. (1965). Diffusion of univalent ions across the lamellae of swollen phospholipid films and the determination of membrane potential. Journal of Molecular Biology, 13(1), 238-252. DOI ↗Chiou, W. L., Riegelman, S. (1971). Pharmaceutical applications of solid dispersions. Journal of Pharmaceutical Sciences, 60(9), 1281-1302. link ↗
Denumiri alternativeliposomal formulation, vesicular delivery, lipid nanoparticlessolid solution, amorphous dispersion, polymer-based formulation
Înrudite33
RezumatLiposomal encapsulation is a formulation technique using lipid bilayer vesicles (liposomes) to enclose drugs, improving bioavailability, reducing toxicity, and enabling targeted delivery. Developed by Alec Bangham in 1965, liposomes are now standard in pharmaceutical development, with several FDA-approved liposomal drugs on the market.Solid dispersion is a formulation technique where a poorly soluble drug is molecularly dispersed in a hydrophilic polymer matrix, improving aqueous solubility and bioavailability. Introduced by Chiou and Riegelman in 1971, solid dispersions remain a key strategy for overcoming solubility-limited absorption.
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ScholarGateCompară metode: Liposome Encapsulation · Solid Dispersion. Preluat la 2026-06-19 de pe https://scholargate.app/ro/compare