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Corelație In Vitro-In Vivo×Cinetică Michaelis-Menten×
DomeniuFarmacologieFarmacologie
FamilieProcess / pipelineProcess / pipeline
Anul apariției19951913
Autorul originalGordon AmidonLeonor Michaelis and Maud Menten
Tipbioavailability predictionmechanistic model
Sursa seminalăAmidon, G. L., Lennernäs, H., Shah, V. P., & Crison, J. R. (1995). A theoretical basis for a biopharmaceutic drug classification: the correlation of in vitro drug product dissolution and in vivo bioavailability. Pharmaceutical Research, 12(3), 413-420. DOI ↗Michaelis, L., & Menten, M. L. (1913). Die Kinetik der Invertinwirkung. Biochemische Zeitschrift, 49, 333-369. link ↗
Denumiri alternativeIVIVCMM kinetics, Michaelis constant, Vmax
Înrudite32
RezumatIVIVC is a mathematical relationship between in vitro and in vivo properties of a drug, developed to predict oral bioavailability from dissolution data. Introduced by Amidon and colleagues in the 1995 Biopharmaceutics Classification System, it bridges laboratory measurements and clinical outcomes to streamline drug development.Michaelis-Menten kinetics describes the rate of enzyme-catalyzed reactions as a function of substrate concentration. Developed by Leonor Michaelis and Maud Menten in 1913, this foundational framework models enzyme catalysis through the rapid-equilibrium approximation and enables prediction of drug metabolism rates in pharmacokinetics.
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ScholarGateCompară metode: In Vitro-In Vivo Correlation · Michaelis-Menten Kinetics. Preluat la 2026-06-19 de pe https://scholargate.app/ro/compare