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Factorul de similaritate f1/f2 pentru dizolvare×Livrarea Medicamentelor Lipozomale×
DomeniuFarmacologieFarmacologie
FamilieProcess / pipelineProcess / pipeline
Anul apariției19961965
Autorul originalJames Moore and Hector FlannerAlec Bangham
Tipsimilarity testingformulation technology
Sursa seminalăMoore, J. W., & Flanner, H. H. (1996). Mathematical comparison of dissolution profiles. Pharmaceutical Technology, 20(6), 64-74. link ↗Bangham, A. D., Standish, M. M., & Watkins, J. C. (1965). Diffusion of univalent ions across the lamellae of swollen phospholipid films and the determination of membrane potential. Journal of Molecular Biology, 13(1), 238-252. DOI ↗
Denumiri alternativef1, f2, similarity factorliposomal formulation, vesicular delivery, lipid nanoparticles
Înrudite33
RezumatThe f1 and f2 factors are dimensionless statistical measures developed by Moore and Flanner to quantify the similarity between two dissolution profiles. Adopted by regulatory agencies (FDA, EMA) as the gold standard for comparing dissolution curves, these factors enable rapid assessment of whether formulation changes significantly impact drug release.Liposomal encapsulation is a formulation technique using lipid bilayer vesicles (liposomes) to enclose drugs, improving bioavailability, reducing toxicity, and enabling targeted delivery. Developed by Alec Bangham in 1965, liposomes are now standard in pharmaceutical development, with several FDA-approved liposomal drugs on the market.
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ScholarGateCompară metode: Dissolution f1/f2 Similarity · Liposome Encapsulation. Preluat la 2026-06-19 de pe https://scholargate.app/ro/compare