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Analīze pēc Šilda (Schild Analysis)×Populācijas farmakodinamiskā modelēšana×
NozareFarmakoloģijaFarmakoloģija
SaimeProcess / pipelineProcess / pipeline
Izcelsmes gads19471992
AutorsHenry SchildLewis Sheiner and Stephen Roush
Tipsantagonism quantificationdose-response modeling
PirmavotsSchild, H. O. (1947). pA, a new scale for the measurement of drug antagonism. Journal of Physiology, 106(3), 337-357. DOI ↗Dahlström, B., & Nyberg, L. (1993). Population pharmacokinetics and pharmacodynamics. Clinical Pharmacokinetics, 24(1), 45-57. link ↗
Citi nosaukumiSchild plot, pA2PopPD, population PD, hierarchical PD modeling
Saistītās33
KopsavilkumsSchild analysis is a quantitative method for characterizing competitive receptor antagonism developed by Henry Schild in 1947. It uses dose-response curves in the presence and absence of antagonist to estimate the antagonist affinity constant (pA2), enabling standardized comparison of antagonist potency across drugs and experimental systems.Population pharmacodynamic (PopPD) modeling integrates pharmacokinetics with individual dose-response relationships across patient populations to characterize drug efficacy and tolerability. Pioneered by Lewis Sheiner and colleagues, PopPD accounts for inter-individual variability in drug effects and enables rational dose optimization and response prediction.
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ScholarGateSalīdzināt metodes: Schild Analysis · Population Pharmacodynamics. Izgūts 2026-06-18 no https://scholargate.app/lv/compare