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Populācijas farmakodinamiskā modelēšana×Fizioloģiski Balstīta Farmakokinētika×
NozareFarmakoloģijaFarmakoloģija
SaimeProcess / pipelineProcess / pipeline
Izcelsmes gads19921997
AutorsLewis Sheiner and Stephen RoushIvan Nestorov
Tipsdose-response modelingpredictive modeling
PirmavotsDahlström, B., & Nyberg, L. (1993). Population pharmacokinetics and pharmacodynamics. Clinical Pharmacokinetics, 24(1), 45-57. link ↗Nestorov, I. (1997). Sensitivity analysis of pharmacokinetic and pharmacodynamic systems. Journal of Pharmacokinetics and Biopharmaceutics, 25(4), 529-543. link ↗
Citi nosaukumiPopPD, population PD, hierarchical PD modelingPBPK, PBPK modeling
Saistītās33
KopsavilkumsPopulation pharmacodynamic (PopPD) modeling integrates pharmacokinetics with individual dose-response relationships across patient populations to characterize drug efficacy and tolerability. Pioneered by Lewis Sheiner and colleagues, PopPD accounts for inter-individual variability in drug effects and enables rational dose optimization and response prediction.PBPK is a mechanistic modeling framework that uses physiological parameters, tissue properties, and drug-specific attributes to predict drug concentration time profiles in the body. Developed rigorously in the 1990s by researchers including Nestorov, PBPK integrates anatomy, biochemistry, and kinetics to enable rational drug development, bridging in vitro data to clinical outcomes.
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ScholarGateSalīdzināt metodes: Population Pharmacodynamics · Physiologically Based Pharmacokinetics. Izgūts 2026-06-19 no https://scholargate.app/lv/compare