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Modellizzazione Farmacodinamica di Popolazione×Analisi di Schild×
CampoFarmacologiaFarmacologia
FamigliaProcess / pipelineProcess / pipeline
Anno di origine19921947
IdeatoreLewis Sheiner and Stephen RoushHenry Schild
Tipodose-response modelingantagonism quantification
Fonte seminaleDahlström, B., & Nyberg, L. (1993). Population pharmacokinetics and pharmacodynamics. Clinical Pharmacokinetics, 24(1), 45-57. link ↗Schild, H. O. (1947). pA, a new scale for the measurement of drug antagonism. Journal of Physiology, 106(3), 337-357. DOI ↗
AliasPopPD, population PD, hierarchical PD modelingSchild plot, pA2
Correlati33
SintesiPopulation pharmacodynamic (PopPD) modeling integrates pharmacokinetics with individual dose-response relationships across patient populations to characterize drug efficacy and tolerability. Pioneered by Lewis Sheiner and colleagues, PopPD accounts for inter-individual variability in drug effects and enables rational dose optimization and response prediction.Schild analysis is a quantitative method for characterizing competitive receptor antagonism developed by Henry Schild in 1947. It uses dose-response curves in the presence and absence of antagonist to estimate the antagonist affinity constant (pA2), enabling standardized comparison of antagonist potency across drugs and experimental systems.
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ScholarGateConfronta i metodi: Population Pharmacodynamics · Schild Analysis. Consultato il 2026-06-18 da https://scholargate.app/it/compare