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Cinetica di Michaelis-Menten×Modellizzazione Farmacodinamica di Popolazione×
CampoFarmacologiaFarmacologia
FamigliaProcess / pipelineProcess / pipeline
Anno di origine19131992
IdeatoreLeonor Michaelis and Maud MentenLewis Sheiner and Stephen Roush
Tipomechanistic modeldose-response modeling
Fonte seminaleMichaelis, L., & Menten, M. L. (1913). Die Kinetik der Invertinwirkung. Biochemische Zeitschrift, 49, 333-369. link ↗Dahlström, B., & Nyberg, L. (1993). Population pharmacokinetics and pharmacodynamics. Clinical Pharmacokinetics, 24(1), 45-57. link ↗
AliasMM kinetics, Michaelis constant, VmaxPopPD, population PD, hierarchical PD modeling
Correlati23
SintesiMichaelis-Menten kinetics describes the rate of enzyme-catalyzed reactions as a function of substrate concentration. Developed by Leonor Michaelis and Maud Menten in 1913, this foundational framework models enzyme catalysis through the rapid-equilibrium approximation and enables prediction of drug metabolism rates in pharmacokinetics.Population pharmacodynamic (PopPD) modeling integrates pharmacokinetics with individual dose-response relationships across patient populations to characterize drug efficacy and tolerability. Pioneered by Lewis Sheiner and colleagues, PopPD accounts for inter-individual variability in drug effects and enables rational dose optimization and response prediction.
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  3. PUBLISHED
  1. v1
  2. 2 Fonti
  3. PUBLISHED

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ScholarGateConfronta i metodi: Michaelis-Menten Kinetics · Population Pharmacodynamics. Consultato il 2026-06-19 da https://scholargate.app/it/compare