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Populationsfarmakodynamisk modellering×Michaelis-Menten-kinetik×
FagområdeFarmakologiFarmakologi
FamilieProcess / pipelineProcess / pipeline
Oprindelsesår19921913
OphavspersonLewis Sheiner and Stephen RoushLeonor Michaelis and Maud Menten
Typedose-response modelingmechanistic model
Oprindelig kildeDahlström, B., & Nyberg, L. (1993). Population pharmacokinetics and pharmacodynamics. Clinical Pharmacokinetics, 24(1), 45-57. link ↗Michaelis, L., & Menten, M. L. (1913). Die Kinetik der Invertinwirkung. Biochemische Zeitschrift, 49, 333-369. link ↗
AliasserPopPD, population PD, hierarchical PD modelingMM kinetics, Michaelis constant, Vmax
Relaterede32
ResuméPopulation pharmacodynamic (PopPD) modeling integrates pharmacokinetics with individual dose-response relationships across patient populations to characterize drug efficacy and tolerability. Pioneered by Lewis Sheiner and colleagues, PopPD accounts for inter-individual variability in drug effects and enables rational dose optimization and response prediction.Michaelis-Menten kinetics describes the rate of enzyme-catalyzed reactions as a function of substrate concentration. Developed by Leonor Michaelis and Maud Menten in 1913, this foundational framework models enzyme catalysis through the rapid-equilibrium approximation and enables prediction of drug metabolism rates in pharmacokinetics.
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ScholarGateSammenlign metoder: Population Pharmacodynamics · Michaelis-Menten Kinetics. Hentet 2026-06-19 fra https://scholargate.app/da/compare