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Cinètica de Michaelis-Menten×Anàlisi de Schild×
CampFarmacologiaFarmacologia
FamíliaProcess / pipelineProcess / pipeline
Any d'origen19131947
Autor originalLeonor Michaelis and Maud MentenHenry Schild
Tipusmechanistic modelantagonism quantification
Font seminalMichaelis, L., & Menten, M. L. (1913). Die Kinetik der Invertinwirkung. Biochemische Zeitschrift, 49, 333-369. link ↗Schild, H. O. (1947). pA, a new scale for the measurement of drug antagonism. Journal of Physiology, 106(3), 337-357. DOI ↗
ÀliesMM kinetics, Michaelis constant, VmaxSchild plot, pA2
Relacionats23
ResumMichaelis-Menten kinetics describes the rate of enzyme-catalyzed reactions as a function of substrate concentration. Developed by Leonor Michaelis and Maud Menten in 1913, this foundational framework models enzyme catalysis through the rapid-equilibrium approximation and enables prediction of drug metabolism rates in pharmacokinetics.Schild analysis is a quantitative method for characterizing competitive receptor antagonism developed by Henry Schild in 1947. It uses dose-response curves in the presence and absence of antagonist to estimate the antagonist affinity constant (pA2), enabling standardized comparison of antagonist potency across drugs and experimental systems.
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ScholarGateCompara mètodes: Michaelis-Menten Kinetics · Schild Analysis. Recuperat el 2026-06-18 de https://scholargate.app/ca/compare