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Factor de similitud de la dissolució f1/f2×Correlació In Vitro-In Vivo×
CampFarmacologiaFarmacologia
FamíliaProcess / pipelineProcess / pipeline
Any d'origen19961995
Autor originalJames Moore and Hector FlannerGordon Amidon
Tipussimilarity testingbioavailability prediction
Font seminalMoore, J. W., & Flanner, H. H. (1996). Mathematical comparison of dissolution profiles. Pharmaceutical Technology, 20(6), 64-74. link ↗Amidon, G. L., Lennernäs, H., Shah, V. P., & Crison, J. R. (1995). A theoretical basis for a biopharmaceutic drug classification: the correlation of in vitro drug product dissolution and in vivo bioavailability. Pharmaceutical Research, 12(3), 413-420. DOI ↗
Àliesf1, f2, similarity factorIVIVC
Relacionats33
ResumThe f1 and f2 factors are dimensionless statistical measures developed by Moore and Flanner to quantify the similarity between two dissolution profiles. Adopted by regulatory agencies (FDA, EMA) as the gold standard for comparing dissolution curves, these factors enable rapid assessment of whether formulation changes significantly impact drug release.IVIVC is a mathematical relationship between in vitro and in vivo properties of a drug, developed to predict oral bioavailability from dissolution data. Introduced by Amidon and colleagues in the 1995 Biopharmaceutics Classification System, it bridges laboratory measurements and clinical outcomes to streamline drug development.
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ScholarGateCompara mètodes: Dissolution f1/f2 Similarity · In Vitro-In Vivo Correlation. Recuperat el 2026-06-20 de https://scholargate.app/ca/compare