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Populationsfarmakodynamisk modellering×Michaelis-Mentens kinetik×
ÄmnesområdeFarmakologiFarmakologi
FamiljProcess / pipelineProcess / pipeline
Ursprungsår19921913
UpphovspersonLewis Sheiner and Stephen RoushLeonor Michaelis and Maud Menten
Typdose-response modelingmechanistic model
UrsprungskällaDahlström, B., & Nyberg, L. (1993). Population pharmacokinetics and pharmacodynamics. Clinical Pharmacokinetics, 24(1), 45-57. link ↗Michaelis, L., & Menten, M. L. (1913). Die Kinetik der Invertinwirkung. Biochemische Zeitschrift, 49, 333-369. link ↗
AliasPopPD, population PD, hierarchical PD modelingMM kinetics, Michaelis constant, Vmax
Närliggande32
SammanfattningPopulation pharmacodynamic (PopPD) modeling integrates pharmacokinetics with individual dose-response relationships across patient populations to characterize drug efficacy and tolerability. Pioneered by Lewis Sheiner and colleagues, PopPD accounts for inter-individual variability in drug effects and enables rational dose optimization and response prediction.Michaelis-Menten kinetics describes the rate of enzyme-catalyzed reactions as a function of substrate concentration. Developed by Leonor Michaelis and Maud Menten in 1913, this foundational framework models enzyme catalysis through the rapid-equilibrium approximation and enables prediction of drug metabolism rates in pharmacokinetics.
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ScholarGateJämför metoder: Population Pharmacodynamics · Michaelis-Menten Kinetics. Hämtad 2026-06-19 från https://scholargate.app/sv/compare