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Pemodelan Farmakodinamik Populasi×Farmakokinetik Berasaskan Fisiologi×
BidangFarmakologiFarmakologi
KeluargaProcess / pipelineProcess / pipeline
Tahun asal19921997
PengasasLewis Sheiner and Stephen RoushIvan Nestorov
Jenisdose-response modelingpredictive modeling
Sumber perintisDahlström, B., & Nyberg, L. (1993). Population pharmacokinetics and pharmacodynamics. Clinical Pharmacokinetics, 24(1), 45-57. link ↗Nestorov, I. (1997). Sensitivity analysis of pharmacokinetic and pharmacodynamic systems. Journal of Pharmacokinetics and Biopharmaceutics, 25(4), 529-543. link ↗
AliasPopPD, population PD, hierarchical PD modelingPBPK, PBPK modeling
Berkaitan33
RingkasanPopulation pharmacodynamic (PopPD) modeling integrates pharmacokinetics with individual dose-response relationships across patient populations to characterize drug efficacy and tolerability. Pioneered by Lewis Sheiner and colleagues, PopPD accounts for inter-individual variability in drug effects and enables rational dose optimization and response prediction.PBPK is a mechanistic modeling framework that uses physiological parameters, tissue properties, and drug-specific attributes to predict drug concentration time profiles in the body. Developed rigorously in the 1990s by researchers including Nestorov, PBPK integrates anatomy, biochemistry, and kinetics to enable rational drug development, bridging in vitro data to clinical outcomes.
ScholarGateSet data
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ScholarGateBandingkan kaedah: Population Pharmacodynamics · Physiologically Based Pharmacokinetics. Dicapai 2026-06-18 daripada https://scholargate.app/ms/compare