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Análisis de Schild×Modelado Farmacodinámico Poblacional×
CampoFarmacologíaFarmacología
FamiliaProcess / pipelineProcess / pipeline
Año de origen19471992
Autor originalHenry SchildLewis Sheiner and Stephen Roush
Tipoantagonism quantificationdose-response modeling
Fuente seminalSchild, H. O. (1947). pA, a new scale for the measurement of drug antagonism. Journal of Physiology, 106(3), 337-357. DOI ↗Dahlström, B., & Nyberg, L. (1993). Population pharmacokinetics and pharmacodynamics. Clinical Pharmacokinetics, 24(1), 45-57. link ↗
AliasSchild plot, pA2PopPD, population PD, hierarchical PD modeling
Relacionados33
ResumenSchild analysis is a quantitative method for characterizing competitive receptor antagonism developed by Henry Schild in 1947. It uses dose-response curves in the presence and absence of antagonist to estimate the antagonist affinity constant (pA2), enabling standardized comparison of antagonist potency across drugs and experimental systems.Population pharmacodynamic (PopPD) modeling integrates pharmacokinetics with individual dose-response relationships across patient populations to characterize drug efficacy and tolerability. Pioneered by Lewis Sheiner and colleagues, PopPD accounts for inter-individual variability in drug effects and enables rational dose optimization and response prediction.
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ScholarGateComparar métodos: Schild Analysis · Population Pharmacodynamics. Recuperado el 2026-06-18 de https://scholargate.app/es/compare