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Análisis de isobologramas×Cinética de Michaelis-Menten×
CampoFarmacologíaFarmacología
FamiliaProcess / pipelineProcess / pipeline
Año de origen19261913
Autor originalSalvatore LoeweLeonor Michaelis and Maud Menten
Tiposynergy quantificationmechanistic model
Fuente seminalLoewe, S. (1926). Die Mischtoxizität. Zeitschrift für Experimentelle Pathologie und Therapie, 24, 315-334. link ↗Michaelis, L., & Menten, M. L. (1913). Die Kinetik der Invertinwirkung. Biochemische Zeitschrift, 49, 333-369. link ↗
Aliasisobol, combination index, synergy testingMM kinetics, Michaelis constant, Vmax
Relacionados32
ResumenIsobologram analysis is a graphical and quantitative method for detecting and classifying drug interactions, developed by Salvatore Loewe in 1926. It uses dose-response data from two drugs applied individually and in combination to determine whether their interaction is additive, synergistic, or antagonistic.Michaelis-Menten kinetics describes the rate of enzyme-catalyzed reactions as a function of substrate concentration. Developed by Leonor Michaelis and Maud Menten in 1913, this foundational framework models enzyme catalysis through the rapid-equilibrium approximation and enables prediction of drug metabolism rates in pharmacokinetics.
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  3. PUBLISHED

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ScholarGateComparar métodos: Isobologram Analysis · Michaelis-Menten Kinetics. Recuperado el 2026-06-20 de https://scholargate.app/es/compare