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Factor de Similitud f1/f2 para Disolución×Entrega de Fármacos Liposomales×
CampoFarmacologíaFarmacología
FamiliaProcess / pipelineProcess / pipeline
Año de origen19961965
Autor originalJames Moore and Hector FlannerAlec Bangham
Tiposimilarity testingformulation technology
Fuente seminalMoore, J. W., & Flanner, H. H. (1996). Mathematical comparison of dissolution profiles. Pharmaceutical Technology, 20(6), 64-74. link ↗Bangham, A. D., Standish, M. M., & Watkins, J. C. (1965). Diffusion of univalent ions across the lamellae of swollen phospholipid films and the determination of membrane potential. Journal of Molecular Biology, 13(1), 238-252. DOI ↗
Aliasf1, f2, similarity factorliposomal formulation, vesicular delivery, lipid nanoparticles
Relacionados33
ResumenThe f1 and f2 factors are dimensionless statistical measures developed by Moore and Flanner to quantify the similarity between two dissolution profiles. Adopted by regulatory agencies (FDA, EMA) as the gold standard for comparing dissolution curves, these factors enable rapid assessment of whether formulation changes significantly impact drug release.Liposomal encapsulation is a formulation technique using lipid bilayer vesicles (liposomes) to enclose drugs, improving bioavailability, reducing toxicity, and enabling targeted delivery. Developed by Alec Bangham in 1965, liposomes are now standard in pharmaceutical development, with several FDA-approved liposomal drugs on the market.
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ScholarGateComparar métodos: Dissolution f1/f2 Similarity · Liposome Encapsulation. Recuperado el 2026-06-19 de https://scholargate.app/es/compare