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Schild-analyse×Populationsfarmakodynamisk modellering×
FagområdeFarmakologiFarmakologi
FamilieProcess / pipelineProcess / pipeline
Oprindelsesår19471992
OphavspersonHenry SchildLewis Sheiner and Stephen Roush
Typeantagonism quantificationdose-response modeling
Oprindelig kildeSchild, H. O. (1947). pA, a new scale for the measurement of drug antagonism. Journal of Physiology, 106(3), 337-357. DOI ↗Dahlström, B., & Nyberg, L. (1993). Population pharmacokinetics and pharmacodynamics. Clinical Pharmacokinetics, 24(1), 45-57. link ↗
AliasserSchild plot, pA2PopPD, population PD, hierarchical PD modeling
Relaterede33
ResuméSchild analysis is a quantitative method for characterizing competitive receptor antagonism developed by Henry Schild in 1947. It uses dose-response curves in the presence and absence of antagonist to estimate the antagonist affinity constant (pA2), enabling standardized comparison of antagonist potency across drugs and experimental systems.Population pharmacodynamic (PopPD) modeling integrates pharmacokinetics with individual dose-response relationships across patient populations to characterize drug efficacy and tolerability. Pioneered by Lewis Sheiner and colleagues, PopPD accounts for inter-individual variability in drug effects and enables rational dose optimization and response prediction.
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ScholarGateSammenlign metoder: Schild Analysis · Population Pharmacodynamics. Hentet 2026-06-18 fra https://scholargate.app/da/compare